Search on: RO 405967 
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Descriptor English:   Mibefradil 
Descriptor Spanish:   Mibefradil 
Descriptor Portuguese:   Mibefradil 
Synonyms English:   Mibefradil Dihydrochloride
Posicor
Ro 40 5967
Ro 40-5967
Ro 405967  
Tree Number:   D02.455.426.559.847.638.960.585
D03.633.100.103.618
D04.615.638.960.585
Definition English:   A benzimidazoyl-substituted tetraline that selectively binds and inhibits CALCIUM CHANNELS, T-TYPE. 
Pharmacological Action:   Antihypertensive Agents
Calcium Channel Blockers
Vasodilator Agents
Cytochrome P-450 CYP1A2 Inhibitors
 
History Note English:   2000; use MIBEFRADIL 1989-1999 
Allowable Qualifiers English:  
AD administration & dosage AE adverse effects
AG agonists AA analogs & derivatives
AN analysis AI antagonists & inhibitors
BL blood CF cerebrospinal fluid
CS chemical synthesis CH chemistry
CL classification EC economics
HI history IM immunology
IP isolation & purification ME metabolism
PK pharmacokinetics PD pharmacology
PO poisoning RE radiation effects
ST standards SD supply & distribution
TU therapeutic use TO toxicity
UR urine  
Record Number:   34398 
Unique Identifier:   D020748 

Occurrence in VHL:
 

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DeCS